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Umbrella Labs
  • Home
    • Sarms for Sale
      • 5-ALPHA-HYDROXY LAXOGENIN for Sale
      • ACP 105 for Sale
      • LGD-4033 for Sale
      • MK-2866 for Sale
      • MK-677 for Sale
      • OTR-AC for Sale
      • RU58841 for Sale
      • S-23 for Sale
      • S-4 for Sale
      • SR-9009 for Sale
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    • Peptides for Sale
      • PEPTIDE LIQUID SPRAY BOTTLE
      • ACE-031 PEPTIDE for Sale
      • ADAMAX PEPTIDE for Sale
      • ADIPOTIDE PEPTIDE for Sale
      • ALPHA MSH PEPTIDE for Sale
      • AOD9604 PEPTIDE for Sale
      • BACTERIOSTATIC WATER for Sale
      • BPC-157 PEPTIDE for Sale
      • CJC-1295 DAC PEPTIDE for Sale
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      • DSIP PEPTIDE for Sale
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      • FOLLISTATIN 344 FST-344 for Sale
      • FRAGMENT 176-191 PEPTIDE for Sale
      • GHK-CU COPPER PEPTIDE for Sale
      • GHRP-2 PEPTIDE (GROWTH HORMONE RELEASING PEPTIDE for Sale
      • VIP PEPTIDE for Sale
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      • PE22.28 PEPTIDE for Sale
      • MOTS-C PEPTIDE for Sale
      • LL-37 PEPTIDE for Sale
      • THYMALIN PEPTIDE for Sale
      • TRIPTORELIN PEPTIDE for Sale
      • SNAP-8 PEPTIDE for Sale
      • TESAMORELIN PEPTIDE for Sale
      • PEG-MGF PEPTIDE for Sale
      • IGF-1 DES PEPTIDE for Sale
      • P21 PEPTIDE LIQUID SPRAY for Sale
      • SERMORELIN PEPTIDE for Sale
      • GONADORELIN PEPTIDE for Sale
      • MELANOTAN II PEPTIDE for Sale
      • HEXARELIN PEPTIDE for Sale
      • MODIFIED GRF (1-29) PEPTIDE for Sale
      • OXYTOCIN PEPTIDE LIQUID SPRAY for Sale
      • SELANK PEPTIDE LIQUID SPRAY for Sale
      • IGF-1 LR3 PEPTIDE for Sale
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    • Nootropics
      • 5-HTP for Sale
      • 7,8-DIHYDROXYFLAVONE HYDRATE (DHT) for Sale
      • 9-ME-BC for Sale
      • ACA for Sale
      • ACETYL L-CARNITINE (ALCAR) for Sale
      • ADRAFINIL for Sale
      • AGOMELATINE for Sale
      • ALPHA-GPC for Sale
      • ANIRACETAM for Sale
      • BEMETHYL for Sale
      • BROMANTANE
      • CB-03-01 for Sale
      • CITICOLINE (CDP-CHOLINE) for Sale
      • COLURACETAM for Sale
      • COMPOUND 7P for Sale
      • D-RIBOSE for Sale
      • PHENYLPIRACETAM for Sale
      • NOOPEPT GVS-111 for Sale
      • FLADRAFINIL (CRL-40,941) for Sale
      • PRAMIRACETAM for Sale
      • TURKESTERONE 20% for Sale
      • PHENYLPIRACETAM HYDRAZIDE for Sale
      • FASORACETAM for Sale
      • NRC NIAGEN for Sale
      • IDRA-21 for Sale
      • SULBUTIAMINE for Sale
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      • URIDINE MONOPHOSPHATE for Sale
      • NSI-189 PHOSPHATE for Sale
      • L-THEANINE for Sale
      • LAXOGENIN for Sale
      • PRL-8-53 for Sale
      • J147 for Sale
      • PHOSPHATIDYLSERINE for Sale
      • NMN (NICOTINAMIDE MONONUCLEOTIDE) for Sale
      • N-ACETYL L-TYROSINE (NALT) for Sale
      • L-TYROSINE for Sale
      • MAGNOLOL 98% MAGNOLIA BARK EXTRACT for Sale
      • KX-826 for Sale
      • WAY 316606 for Sale
      • N-PHENETHYL DIMETHYLAMINE (10 GRAMS) for Sale
      • NEFIRACETAM for Sale
      • VINPOCETINE for Sale
    • Lab Supplies
      • 1mL Pipette Dropper for Sale
      • 6mg – 10mg Micro Scoop for Sale
      • 10mg – 15mg Micro Scoop for Sale
      • 25mg – 30mg Micro Scoop for Sale
      • 150mg Micro Scoop for Sale
      • 30mL (1oz) Glass Bottle for Sale
      • 30mL Bottle w 1mL Dropper for Sale
      • 500mg (0.5g) Micro Scoop for Sale
      • Micro Scoops Variety Pack for Sale
    • Research Chemicals for Sale
      • RU58841 SOLUTION (SARM SUPPORT) for Sale
      • RU58841 POWDER (SARM SUPPORT) for Sale
  • More
    • Home
      • Sarms for Sale
        • 5-ALPHA-HYDROXY LAXOGENIN for Sale
        • ACP 105 for Sale
        • LGD-4033 for Sale
        • MK-2866 for Sale
        • MK-677 for Sale
        • OTR-AC for Sale
        • RU58841 for Sale
        • S-23 for Sale
        • S-4 for Sale
        • SR-9009 for Sale
        • SR-9011 for Sale
        • YK-11 for Sale
        • GW 0742 for Sale
        • RAD-140 for Sale
        • GW-501516 for sale
        • RAD-150 for Sale
        • LGD-3303 for Sale
      • Peptides for Sale
        • PEPTIDE LIQUID SPRAY BOTTLE
        • ACE-031 PEPTIDE for Sale
        • ADAMAX PEPTIDE for Sale
        • ADIPOTIDE PEPTIDE for Sale
        • ALPHA MSH PEPTIDE for Sale
        • AOD9604 PEPTIDE for Sale
        • BACTERIOSTATIC WATER for Sale
        • BPC-157 PEPTIDE for Sale
        • CJC-1295 DAC PEPTIDE for Sale
        • CJC-1295 NO DAC PEPTIDE for Sale
        • DSIP PEPTIDE for Sale
        • EPITALON PEPTIDE for Sale
        • FOLLISTATIN 344 FST-344 for Sale
        • FRAGMENT 176-191 PEPTIDE for Sale
        • GHK-CU COPPER PEPTIDE for Sale
        • GHRP-2 PEPTIDE (GROWTH HORMONE RELEASING PEPTIDE for Sale
        • VIP PEPTIDE for Sale
        • KPV PEPTIDE for Sale
        • PE22.28 PEPTIDE for Sale
        • MOTS-C PEPTIDE for Sale
        • LL-37 PEPTIDE for Sale
        • THYMALIN PEPTIDE for Sale
        • TRIPTORELIN PEPTIDE for Sale
        • SNAP-8 PEPTIDE for Sale
        • TESAMORELIN PEPTIDE for Sale
        • PEG-MGF PEPTIDE for Sale
        • IGF-1 DES PEPTIDE for Sale
        • P21 PEPTIDE LIQUID SPRAY for Sale
        • SERMORELIN PEPTIDE for Sale
        • GONADORELIN PEPTIDE for Sale
        • MELANOTAN II PEPTIDE for Sale
        • HEXARELIN PEPTIDE for Sale
        • MODIFIED GRF (1-29) PEPTIDE for Sale
        • OXYTOCIN PEPTIDE LIQUID SPRAY for Sale
        • SELANK PEPTIDE LIQUID SPRAY for Sale
        • IGF-1 LR3 PEPTIDE for Sale
        • SEMAX PEPTIDE LIQUID SPRAY for Sale
        • GHRP-6 PEPTIDE (GROWTH HORMONE RELEASING PEPTIDE 6) for Sale
        • IPAMORELIN PEPTIDE for Sale
        • MGF MECHANO GROWTH FACTOR PEPTIDE for Sale
        • PT-141 BREMELANOTIDE PEPTIDE for Sale
        • TB-500 THYMOSIN BETA-4 PEPTIDE for Sale
      • Nootropics
        • 5-HTP for Sale
        • 7,8-DIHYDROXYFLAVONE HYDRATE (DHT) for Sale
        • 9-ME-BC for Sale
        • ACA for Sale
        • ACETYL L-CARNITINE (ALCAR) for Sale
        • ADRAFINIL for Sale
        • AGOMELATINE for Sale
        • ALPHA-GPC for Sale
        • ANIRACETAM for Sale
        • BEMETHYL for Sale
        • BROMANTANE
        • CB-03-01 for Sale
        • CITICOLINE (CDP-CHOLINE) for Sale
        • COLURACETAM for Sale
        • COMPOUND 7P for Sale
        • D-RIBOSE for Sale
        • PHENYLPIRACETAM for Sale
        • NOOPEPT GVS-111 for Sale
        • FLADRAFINIL (CRL-40,941) for Sale
        • PRAMIRACETAM for Sale
        • TURKESTERONE 20% for Sale
        • PHENYLPIRACETAM HYDRAZIDE for Sale
        • FASORACETAM for Sale
        • NRC NIAGEN for Sale
        • IDRA-21 for Sale
        • SULBUTIAMINE for Sale
        • SPERMIDINE 3HCL for Sale
        • URIDINE MONOPHOSPHATE for Sale
        • NSI-189 PHOSPHATE for Sale
        • L-THEANINE for Sale
        • LAXOGENIN for Sale
        • PRL-8-53 for Sale
        • J147 for Sale
        • PHOSPHATIDYLSERINE for Sale
        • NMN (NICOTINAMIDE MONONUCLEOTIDE) for Sale
        • N-ACETYL L-TYROSINE (NALT) for Sale
        • L-TYROSINE for Sale
        • MAGNOLOL 98% MAGNOLIA BARK EXTRACT for Sale
        • KX-826 for Sale
        • WAY 316606 for Sale
        • N-PHENETHYL DIMETHYLAMINE (10 GRAMS) for Sale
        • NEFIRACETAM for Sale
        • VINPOCETINE for Sale
      • Lab Supplies
        • 1mL Pipette Dropper for Sale
        • 6mg – 10mg Micro Scoop for Sale
        • 10mg – 15mg Micro Scoop for Sale
        • 25mg – 30mg Micro Scoop for Sale
        • 150mg Micro Scoop for Sale
        • 30mL (1oz) Glass Bottle for Sale
        • 30mL Bottle w 1mL Dropper for Sale
        • 500mg (0.5g) Micro Scoop for Sale
        • Micro Scoops Variety Pack for Sale
      • Research Chemicals for Sale
        • RU58841 SOLUTION (SARM SUPPORT) for Sale
        • RU58841 POWDER (SARM SUPPORT) for Sale

RAD-140 for Sale

RAD 140 Effects on Animal Body Mass

RAD 140 SARM, or (2-chloro-4-[[(1R,2S)-1-[5-(4-cyanophenyl)-1,3,4-oxadiazol-2-yl]-2-hydroxypropyl]amino]-3-methylbenzonitrile, also known as testolone was originally synthesized for Radius Health Inc. in conjunction with researchers from the University of Illinois, Obiter Research, and Cambridge Major Laboratories.

Per the initial paper detailing the synthesis and preliminary findings of the compound, RAD140 has the stability to (t1/2 >2 h) in incubations with rat and monkey microsomes, as well as a high affinity for the androgen receptor (Ki = 7 nM), approximately 4 times the affinity than that of testosterone itself. At the same time, the nearest hormone receptor activated by RAD140 was progesterone at a level of 750nM.

The earliest primate studies on RAD-140 indicated that even at the lowest dose range 0.1mg/kg, juvenile macaques gained a mean of ten percent in body weight, during the 28-day trial period, which was primarily confirmed to be lean body mass via DEXA scans performed before and after the trial period, however, this was somewhat variable.

RAD 140 Effects on Neurons

In a study conducted by Jayaraman et. Al, gonadectomized, male rats were studied to see the effects supplementation with RAD 140 had in regards to neuroprotection in order to make conclusions regarding the usefulness of SARMs against neurodegenerative disorders.

The rats were orally provided with 1 mg/kg a day of RAD 140 for 2 weeks. It was found that RAD140 was able to reduce apoptosis caused by Aᵝ, apoptosis activator II, and hydrogen peroxide by a significant amount. This is due to the role MAPK signaling plays in neuroprotection.

Aᵝ was by far the most potent of the apoptosis insults introduced to the rats. After 24 hours of exposure to Aᵝ, 50% of viable neurons in the rats had decreased, however, when given RAD 140 in a concentration-dependent matter, the viability of the neurons had increased exponentially. The most effective concentration of RAD 140 was 100 nM, which led to approximately 90% neuron survival after Aᵝ exposure (https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3959610/).

In addition to measuring the neuroprotection against various apoptosis insults, researchers also measured the effects RAD 140 had on kainate-induced neuron death. It was found that when compared to treatment with a vehicle, kainate-induced neuron death was significantly reduced (https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3959610/).

Our compounds are available in powdered, poly-cell, and standard polyethylene glycol formulations. We employ an amphiphilic copolymer to form polymeric micelles that enhance the bioavailability of select SARMs In animal models.

Furthermore, our nano-emulsification process ensures minimum polymeric micelle size and variance. Most importantly, our Poly-Cell FormulaTM is optimized for sublingual absorption with a minimal taste profile. This stands in contrast to PEG, which is often intolerable for sublingual delivery due to its very unpleasant taste, leading to poor compliance among research participants. However, we do offer PEG for researchers who prefer the standard research delivery method.

The primary concern for SARM researchers today is product purity. Umbrella Labs insures and guarantees its product purity by incorporating a process of Independent testing using Mass Spectrometry and Ultraviolet Radiation. Certificates of our product Independent tests are posted with our product descriptions. Not only are our products guaranteed pure, but they are also guaranteed to be accurately concentrated as well.

**LAB USE ONLY**

*This information is for educational purposes only and does not constitute medical advice. THE PRODUCTS DESCRIBED HEREIN ARE FOR RESEARCH USE ONLY. All clinical research must be conducted with oversight from the appropriate Institutional Review Board (IRB). All preclinical research must be conducted with oversight from the appropriate Institutional Animal Care and Use Committee (IACUC) following the guidelines of the Animal Welfare Act (AWA).


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