2006-2010
33 - Poly-heteroaryl derivatives for the treatment of cancer.
Chi-Hung Nguyen, Myriam Rouchon Dagois, Aurore Guédin-Beaurepaire, David Monchaud, Marie-Paule Teulade-Fichou, Jean-Francois Riou, Jean-Louis Mergny, David Grierson,
32 - “One ring to bind them all” – Part I: The efficiency of the macrocyclic scaffold for G-quadruplex DNA recognition
David Monchaud, Anton Granzhan, Nicolas Saettel, Aurore Guédin, Jean-Louis Mergny, Marie-Paule Teulade-Fichou
J. Nucleic Acids, 2010, 2010, ID460561.
31 - “One ring to bind them all” – Part II: Identification of Promising G-Quadruplex Ligands by Screening of Cyclophane-type Macrocycles.
Anton Granzhan, David Monchaud, Nicolas Saettel, Aurore Guédin, Jean-Louis Mergny, and Marie-Paule Teulade-Fichou
J. Nucleic Acids, 2010, 2010, ID525862.
30 - Template-Assembled Synthetic G-Quadruplex (TASQ): A Useful System for Investigating the Interactions of Ligands with Constrained Quadruplex Topologies.
Pierre Murat, Romaric Bonnet, Agéline Van der Heyden, Nicolas Spinelli, Pierre Labbé, David Monchaud, Marie-Paule Teulade-Fichou, Pascal Dumy, Eric Defrancq
Chem. Eur. J., 2010, 16, 6106.
29 - G4-FID: a fluorescent DNA probe displacement assay for rapid evaluation of quadruplex ligands.
David Monchaud, Marie-Paule Teulade-Fichou
in "G-Quadruplex DNA: Methods and Protocols", P. Baumann (Ed.)
Meth. Mol. Biol., 2010, 608, 257-271.
28 - Synthesis and evaluation of fused bispyrimidinoacridines as novel pentacyclic analogues of quadruplex-binders BRACO-19.
Julien Debray, Walid Zeghida, Muriel Jourdan, David Monchaud, Marie-Louise Dheu-Andries, Pascal Dumy, Marie-Paule Teulade-Fichou, Martine Demeunynck
Org. Biomol. Chem., 2009, 7, 5219-5228.
27 - Exclusive platination of loop adenines in the human telomeric G-quadruplex.
Hélène Bertrand, Sophie Bombard, David Monchaud, Eric Talbot, Aurore Guedin, Jean-Louis Mergny, Renate Grünter, Patrick J. Bednarski, Marie-Paule Teulade-Fichou
Org. Biomol. Chem., 2009, 7, 2864-2871.
26 - Engineering bisquinolinium/thiazole orange conjugates for fluorescent sensing of G-quadruplex DNA.
Peng Yang, Anne De Cian, Marie-Paule Teulade-Fichou, Jean-Louis Mergny, David Monchaud
Angew. Chem. Int. Ed., 2009, 48, 2188-2191
25 - New platinum(II) complexes targeting the loops of the human telomeric G-quadruplex.
Hélène Bertrand, Sophie Bombard, David Monchaud, Marie-Paule Teulade-Fichou
Nucleic Acids Symp. Ser., 2008, 52, 163-164
24 - Ligands playing musical chairs with G-quadruplex DNA: A rapid and simple displacement assay for identifying selective G-quadruplex binders.
David Monchaud, Clémence Allain, Hélène Bertrand, Nicolas Smargiasso, Frédéric Rosu, Valérie Gabelica, Anne De Cian, Jean-Louis Mergny, Marie-Paule Teulade-Fichou
Biochimie, 2008, 90, 1207-1223
23 - A hitchhiker's guide to G-quadruplex ligands
David Monchaud, Marie-Paule Teulade-Fichou
Org. Biomol. Chem., 2008, 4, 627-636
→ In the 25 most cited articles in ISI Web of knowledge (entry "quadruplex") out of >4100 references!
22 - A Metal-Mediated Conformational Switch Controls G-Quadruplex Binding Affinity.
David Monchaud, Peng Yang, Laurent Lacroix, Marie-Paule Teulade-Fichou, Jean-Louis Mergny
Angew. Chem. Int. Ed., 2008, 47, 4858-4861
21 - Plasmodium Telomeric Sequences: Structure, Stability and Quadruplex Targeting by Small Compounds.
Anne De Cian, Philippe Grellier, Elisabeth Mouray, Delphine Depoix, Hélène Bertrand, David Monchaud, Marie-Paule Teulade-Fichou, Jean-Louis Mergny, Patrizia Alberti
ChemBioChem, 2008, 9, 2730-2739
20 - Inhibition of Dicing of Guanosine-Rich shRNAs by Quadruplex-Binding Compounds.
Anja Henn, Astrid Joachimi, Diana P. N. Gonçalves, David Monchaud, Marie-Paule Teulade-Fichou, Jeremy K. M. Sanders, Jörg S. Hartig
ChemBioChem, 2008, 9, 2722-2729
19 - The importance of metal geometry in the recognition of G-quadruplex-DNA by metal-terpyridine complexes.
Hélène Bertrand, David Monchaud, Anne De Cian, Régis Guillot, Jean-Louis Mergny and Marie-Paule Teulade-Fichou
Org. Biomol. Chem., 2007, 5, 2555-2559
18 - A platinum-quinacridine hybrid as a G-quadruplex ligand.
Hélène Bertrand, Sophie Bombard, David Monchaud and Marie-Paule Teulade-Fichou
J. Biol. Inorg. Chem., 2007, 12, 1003-1014
17 - Thiazole Orange: A Useful Probe for Fluorescence Sensing of G-Quadruplex-Ligand Interactions.
David Monchaud, Clémence Allain, Marie -Paule Teulade-Fichou
Nucleosides, Nucleotides Nucleic Acids, 2007, 26, 1585-1588
16 - G-Quadruplex Recognition by Quinacridines: a SAR, NMR, and Biological Study.
Candide Hounsou, Lionel Guittat, David Monchaud, Muriel Jourdan, Nicolas Saettel, Jean-Louis Mergny, Marie-Paule Teulade-Fichou
15 - Reevaluation of telomerase inhibition by quadruplex ligands and their mechanisms of action.
Anne De Cian, Gael Cristofari, Patrick Reichenbach, Elsa De Lemos, David Monchaud, Marie-Paule Teulade-Fichou, Kazuo Shin-ya, Laurent Lacroix, Joachim Lingner, Jean-Louis Mergny
Proc. Natl. Acad. Sci. USA, 2007, 104, 17347-17352
14 - Highly Efficient G-Quadruplex Recognition by Bisquinolinium Compounds.
Anne De Cian, Elsa DeLemos, Jean-Louis Mergny, Marie-Paule Teulade-Fichou, and David Monchaud
J. Am. Chem. Soc. , 2007, 129, 1856-1857
13 - Beneficial Effect of Mukaiyama Reagent on Macrobislactamization Reactions.
Lucie Vandromme, David Monchaud, Marie-Paule Teulade-Fichou
12 - Development of a fluorescent intercalator displacement assay (G4-FID) for establishing quadruplex-DNA affinity and selectivity of putative ligands.
David Monchaud, Clémence Allain, Marie-Paule Teulade-Fichou
Bioorg. Med. Chem. Lett., 2006, 16, 4842-4845
11 - FRET Templated by G-Quadruplex DNA: A Specific Ternary Interaction Using an Original Pair of Donor/Acceptor Partners.
Clémence Allain, David Monchaud, and Marie-Paule Teulade-Fichou
J. Am. Chem. Soc., 2006, 128, 11890-11893