Publications

Oral 18-methoxycoronaridine activity in simian and murine Leishmania amazonensis infection. Frontiers in Pharmacology, 1-16.

Structure-Based Discovery of Selective Vaccinia-Related Kinase 1 Inhibitors and Fluorogenic Active-Site Probes. Journal of Biological Chemistry, 111355.

How to Perform a Tracer Displacement BRET Assay for the TRPML1 Ion Channel. Bio-protocol, 1.

Synthesis of 6-Arylaminoflavones via Buchwald–Hartwig Amination and Its Anti-Tumor Investigation. Reactions, 6 (42), 1.

Fragment Screening by Weak Affinity Chromatography Identifies Ligands for Neisseria gonorrhoeae Undecaprenyl Diphosphate Synthase. bioRvix.

Discovery of pyrazolo [3, 4-d] pyrimidines as novel mitogen-activated protein kinase kinase 3 (MKK3) inhibitors. Bioorganic and Medicinal Chemistry, 98, 117561.

Novel Dihydropteridinone Derivatives As Potent Inhibitors of the Understudied Human Kinases Vaccinia-Related Kinase 1 and Casein Kinase 1δ/ε. Journal of Medicinal Chemistry, 67 (11), 8609.

Rational Exploration of 2,4-Diaminopyrimidines as DHFR Inhibitors Active against Mycobacterium abscessus and Mycobacterium avium, Two Emerging Human Pathogens. Journal of Medicinal Chemistry, 67 (21), 19143.

(S)‐ML‐SA1 Activates Autophagy via TRPML1‐TFEB Pathway. ChemBioChem, 25 (12), e202400506.

A novel BRET-based assay to investigate binding and residence time of unmodified ligands to the human lysosomal ion channel TRPML1 in intact cells. Journal of Biological Chemistry, 299 (6), 104807.