Binding and internalisation inhibitors
7-hydroxystaurosporine
Aclidinium
Afeletecan
Alprostadil
Amcinonide
Amiodarone
Apilimod
Aprepitant
Atropine
Azathioprine
AZD-8330
Azilsartan
Bafetinib
Barusiban
Bekanamycin
Bemcentinib
Bendamustine
Berzosertib
Bicalutamide
Birinapant
Brigatinib
Brilacidin
Bromocriptine
Brompheniramine
Bunazosin
Calcifediol
Camostat
Captopril
Cefixime
Ceritinib
Cimicoxib
Clobazam
Cobimetinib
Conivaptan
Copanlisib
CP-195543
Dacomitinib
Dasatinib
Decanoyl-RVKR-chloromethylketone
Deferasirox
Delavirdine
Desvenlafaxine
Deutivacaftor
Dihydroergotamine
Diminazene
Disopyramide
Doxazosin
Dutasteride
Elamipretide
Eletriptan
Entrectinib
Enzalutamide
Fenofibrate
Fluvastatin
Gentamicin
Iloprost
Ipamorelin
Isocarboxazid
Kanamycin
Ketoconazole
Lapatinib
Levomefolate
Lixivaptan
Lometrexol
Lomibuvir
Lumacaftor
MDL-28170
Megestrol acetate
Methsuximide
Methylnaltrexone
MG-132
MI-1851
MI-1900
MI-432
Midazolam
Modithromycin
Nafamostat
Nafithromycin
Naloxone
Naphthofluorescein
Nebivolol
Netilmicin
Netupitant
Nilotinib
Nilutamide
Nimesulide
Omeprazole
ONO 5334
Orphenadrine
Otamixaban
Panobinostat
Pelitinib
Pelitrexol
Perphenazine
Pimecrolimus
Pioglitazone
Pramoxine
Prazosin
Primaquine
Prochlorperazine
Propylhexedrine
Proxalutamide
Rabeprazole
Raltitrexed
Rebamipide
Recoflavone
Ruzasvir
Sivifene
Sonidegib
Spironolactone
Tadalafil
Terazosin
Tetrahydroquinoline oxocarbazate
Ticlopidine
Tivozanib
Treprostinil
Triazolam
Umifenovir
Vadimezan
VBY-825
Zileuton
Ziritaxestat