Binding and internalisation inhibitors

7-hydroxystaurosporine

Aclidinium

Afeletecan

Alprostadil

Amcinonide

Amiodarone

Apilimod

Aprepitant

Atropine

Azathioprine

AZD-8330

Azilsartan

Bafetinib

Barusiban

Bekanamycin

Bemcentinib

Bendamustine

Berzosertib

Bicalutamide

Birinapant

Brigatinib

Brilacidin

Bromocriptine

Brompheniramine

Bunazosin

Calcifediol

Camostat 

Captopril

Cefixime

Ceritinib

Cimicoxib

Clobazam

Cobimetinib

Conivaptan

Copanlisib

CP-195543

Dacomitinib

Dasatinib

Decanoyl-RVKR-chloromethylketone

Deferasirox

Delavirdine

Desvenlafaxine

Deutivacaftor

Dihydroergotamine

Diminazene

Disopyramide

Doxazosin

Dutasteride

Elamipretide

Eletriptan

Entrectinib

Enzalutamide 

Fenofibrate

Fluvastatin

Gentamicin

Iloprost

Ipamorelin

Isocarboxazid

Kanamycin

Ketoconazole

Lapatinib

Levomefolate

Lixivaptan

Lometrexol

Lomibuvir

Lumacaftor

MDL-28170

Megestrol acetate

Methsuximide



Methylnaltrexone

MG-132

MI-1851

MI-1900

MI-432

Midazolam

Modithromycin

Nafamostat

Nafithromycin

Naloxone

Naphthofluorescein

Nebivolol

Netilmicin

Netupitant

Nilotinib

Nilutamide

Nimesulide

Omeprazole

ONO 5334

Orphenadrine

Otamixaban

Panobinostat

Pelitinib

Pelitrexol

Perphenazine

Pimecrolimus

Pioglitazone

Pramoxine

Prazosin

Primaquine

Prochlorperazine

Propylhexedrine

Proxalutamide

Rabeprazole

Raltitrexed

Rebamipide

Recoflavone

Ruzasvir

Sivifene

Sonidegib

Spironolactone

Tadalafil

Terazosin

Tetrahydroquinoline oxocarbazate 

Ticlopidine

Tivozanib

Treprostinil

Triazolam

Umifenovir 

Vadimezan

VBY-825

Zileuton

Ziritaxestat