1.          Taewoo Kim, Shin-Yae Choi, Hee-Won Bae, Hyun Su Kim, Hoon Jeon, Haejun Oh, Sung-Hoon Ahn, Jongkook Lee, Young-Ger Suh, You-Hee Cho,* Seok-Ho Kim,* Design, synthesis, and evaluation of N1,N3-dialkyldioxonaphthoimidazoliums as antibacterial agents against methicillin-resistant Staphylococcus aureus, Eur. J. Med. Chem. 2024, 272, 116454. (2024-06-05)

2.         Ji Hyun Lee, Hyeon Joo Ham, Hye-Min Bae, Kyoung-Moon Han, Jongkook Lee, Hyung Il Kim,* Establishment of high-performance liquid chromatography-photodiode array method for 43 weight loss agents and effect of basic environment on bisacodyl degradation, Rapid Commun. Mass. Spectrom. 2024, 38, e9705. (2024-03-15)

3.          Duy-Viet Vo, Jongkook Lee, Haeil Park,* 1,2,3-Triazole analogs with bulky and conformationally rigid substructures: Synthesis and in vitro evaluation as DPP-4 inhibitors, Bull. Korean Chem. Soc. 2023, 44, 425–428. (2023-05)

4.         Taewoo Kim, Hyun Su Kim, Jaebong Jang, Dong-Jun Kim, Jongkook Lee, Dongjoo Lee,* Seok-Ho Kim,* Synthesis of 7,20-Dihydroxy-4’,5’-Dimethoxyisoflavanone, a Phytoestrogen with Derma Papilla Cell Proliferative Activity, Molecules 2022, 27, 6660. (2022-10-07)

5.    Hyo Jeong Lee, Yeongyu Moon, Jungil Choi, Jeong Doo Heo, Sekwang Kim, Hari Krishna Nallapaneni, Young-Won Chin, Jongkook Lee, Sun-Young Han,* Characterization of KRC-108 as a TrkA Kinase Inhibitor with Anti-Tumor Effects, Biomol. Ther. 2022, 30, 360–367. (2022-07)

6.          Ji Hyun Lee,¶ Ji Hye Han,¶ Hyeon Joo Ham, Hyungil Kim, Jongkook Lee, Sun Young Baek,* Development of a method for simultaneous screening of four natural derived steroids and their analogues used as dietary supplements via liquid chromatography-quadrupole-time of flight mass spectrometry and liquid chromatography-tandem mass spectrometry, Food Addit. Contam. Part A Chem. Anal. Control Expo. Risk Assess. 2022, 39, 829–837. (2022-05)

7.        Thien Nhan Lu, Minjung Kwak, Mallesham Samala, Minji Son, Jungjoong Hwang, Suresh Mandava, Thuy Trang Pham, Haeil Park, Hyoungsu Kim, Deukjoon Kim, Jongkook Lee,* Highly Stereoselective Asymmetric Total Synthesis of (−)-Jimenezin via Sequential Intramolecular Amide Enolate Alkylation, Org. Lett. 2022, 24, 1652−1656. (2022-03-04)

8.           Chung Hwan Hong,¶ Myoung Seok Ko,¶ Jae Hyun Kim,¶ Hyunkyung Cho, Chi-Ho Lee, Ji Eun Yoon, Ji-Young Yun, In-Jeoung Baek, Jung Eun Jang, Seung Eun Lee, Yun Kyung Cho, Ji Yeon Baek, Soo Jin Oh, Bong Yong Lee, Joon Seo Lim, Jongkook Lee, Sean M. Hartig, Laura Conde de la Rosa, Carmen Garcia-Ruiz, Ki-Up Lee, Jose C. Fernández-Checa,* Ji Woong Choi,* Sanghee Kim,* Eun Hee Koh,* Sphingosine 1-Phosphate Receptor 4 Promotes Nonalcoholic Steatohepatitis by Activating NLRP3 Inflammasome, Cell. Mol. Gastroenterol. Hepatol. 2022, 13, 925–947. (2022-01-01)

9.           Ji Hyun Lee, Ji Hye Han, Eun-Ju Jung, Hari Krishna Nallapaneni, Nam Sook Kim, Jongkook Lee, Sun Young Baek,* Food Addit. Contam. Part A Chem. Anal. Control Expo. Risk Assess. 2021, 38, 1075–1086. (2021-07)

10.        Duy-Viet Vo, Kwon Ho Hong, Jongkook Lee, Haeil Park,* Synthesis, in vitro evaluation, and computational simulations studies of 1,2,3-triazole analogues as DPP-4 inhibitors, Bioorg. Med. Chem. 2021, 29, 115861. (2021-01)

11.           Jungjoong Hwang, Insuk Song, Kwangho Lee, Hyoung Rae Kim, Eun-Hye Hong, Jung Soon Hwang, Sung-Hoon Ahn, Jongkook Lee,* KRCA-0008 suppresses ALK-positive anaplastic large-cell lymphoma growth, Invest. New Drugs 2020, 38, 1282–1291. (2020-10)

12.      Kandasamy Saravanakumar, Suresh Mandava, Ramachandran Chellia, Elango Jeevithan, Ravi Shankar Babu Yelamanchi, Deepthi Mandava, Wu Wen-Hui, Jongkook Lee, Deog-Hwan Oh, Kandasamy Kathiresanf, Myeong-Hyeon Wang,* Novel metabolites from Trichoderma atroviride against human prostate cancer cells and their inhibitory effect on Helicobacter pylori and Shigella toxin producing Escherichia coli, Microb.l Pathog. 2019, 126, 19–26. (2019-01)

13.       Seon-Hyeong Lee, Won-Kyu Lee, Nayeon Kim, Joon Hee Kang, Kyung-Hee Kim, Seul-Gi Kim, Jae-Seon Lee, Soohyun Lee, Jongkook Lee, Jungnam Joo, Woo Sun Kwon, Sun Young Rha, Soo-Youl Kim,* Renal Cell Carcinoma Is Abrogated by p53 Stabilization through Transglutaminase 2 Inhibition, Cancers, 2018, 10, 455 (18 pages). (2018-11-19)

14.          Ji Hyun Lee, Han Na Park, Aeran Jung, Suresh Mandava, Seongsoo Park, Jongkook Lee,* Hoil Kang,* Isolation and characterisation of a novel sildenafil analogue adulterant,desmethylpiperazinyl propoxysildenafil, in a dietary supplement, Sci. Justice 2018, 58, 447–454. (2018-11)

15.         Jae-Hyoung Song, Aeri Shim, Yeon-Jeong Kim, Jae-Hee Ahn, Bo-Eun Kwon, Thuy Trang Pham, Jongkook Lee, Sun-Young Chang, Hyun-Jeong Ko,* Antiviral and Anti-Inflammatory Activities of Pochonin D, a Heat Shock Protein 90 Inhibitor, against Rhinovirus Infection, Biomol. Ther. 2018, 26, 576-583. (2018-11-01) 

16.           Mallesham Samala,  Thien Nhan Lu, Suresh Mandava, Jungjoong Hwang, Ganganna Bogonda, Donghoon Kim, Haeil Park, Deukjoon Kim, Jongkook Lee,* Stereoselective Protection-Free Asymmetric Total Synthesis of (+)-Chamuvarinin, a Potent Anticancer and Antitrypanosomal Agent: Substrate-Controlled Construction of the Adjacently Linked Oxatricyclic Core by Internal Alkylation, Org. Lett. 2018, 20, 6398-6402. (2018-10-19)

17.     Momna Rub, Ramachandran Chellia, Kandasamy Saravanakumar, Suresh Mandava, Imran Khan, Charles Nkufi Tango, Mohammad Shakhawat Hussain, Eric Banan-Mwine Daliri, Se-Hun Kim, Sudha Rani Ramakrishnan, Myeong-Hyeon Wang, Jongkook Lee, Joong-Ho Kwon, Sangeeta Chandrashekar, Deog-Hwan Oh, Preservative effect of Chinese cabbage (Brassica rapa subsp. pekinensis) extract on their molecular docking, antioxidant and antimicrobial properties, PloS One 2018, 13, e0203306. (2018-10-03)

18.         Ji Hyun Lee, Aeran Jung, Han Na Park, Changhee Lee, Suresh Mandava, Sung-jun Lim, Byoung-bok Lim, Sung-Kwan Park, Jongkook Lee,* Hoil Kang,* Identification and characterization of an indazole-3-carboxamide class synthetic cannabinoid: 2-[1-(cyclohexylmethyl)-1H-indazole-3-carboxamido]-3,3-dimethylbutanoic acid (DMBA-CHMINACA), Forensic Sci. Int. 2018, 291, 167–174. (2018-10-01)

19.         Sungjin Ahn, Moonyoung Lee, Seungchan An, Sooyeol Hyun, Jiho Hwang, Jongkook Lee,* Minsoo Noh,* 2-Formyl-komarovicine promotes adiponectin production in human mesenchymal stem cells through PPARγ partial agonism, Bioorg. Med. Chem. 2018, 26, 1069–1075. (2018-03-01)

20.      Jungjoong Hwang, Jiho Hwang, Bogonda Ganganna, Insuk Song, Moon Young Heo, Sung‑Hoon Ahn, Jongkook Lee,* Metabolic and pharmacokinetic characterization of a new synthetic cannabinoid APINAC in rats, Forensic Toxicol. 2018, 36, 88–101. (2018-01)

21.         Ji Hyun Lee, Han Na Park, Hyoung Joon Park, Nam Sook Kim, Sung-Kwan Park, Jongkook Lee,* Sun Young Baek,* Isolation and structural identification of a novel minoxidil analogue in an illegal dietary supplement: triaminodil, Food Addit. Contam. Part A Chem. Anal. Control Expo. Risk Assess. 2018, 35, 2–9. (2018-01)

22.        Hyeonjeong Choe, Hyukjoon Cho, Hyun-Jeong Ko, Jongkook Lee,* Total Synthesis of (+)-Pochonin D and (+)-Monocillin II via Chemo- and Regioselective Intramolecular Nitrile Oxide Cycloaddition, Org. Lett. 2017, 19, 6004–6007. (2017-11-03)

23.       Thien Nhan Lu,* Bogonda Ganganna, Thuy Trang Pham, Anh Van Vo, Thien Phuc Lu, Huong-Giang Thi Nguyen, My-Nuong Thi Nguyen, Phuong Nguyen Huynh, Ngoc Tuyen Truong, Jongkook Lee, Antitumor effect of the integrin a4 signaling inhibitor JK273 in non-small cell lung cancer NCI-H460 cells, Biochem. Biophys. Res. Commun. 2017, 491, 355–360. (2017-09-16)

24.       Bogonda Ganganna, Thien Nhan Lu, Jiho Hwang, Jungjoong Hwang, Suresh Mandava, Yoonchang Jang, Mallesham Samala, Haeil Park, Jongkook Lee,* First Syntheses of (±)-Butesuperins A and B, Bull. Korean Chem. Soc. 2017, 38, 944–947. (2017-08)

25.         Jung-Ah Do, Eunyoung Noh, Soon-Byung Yoon, Ji Hyun Lee, Sung-Kwan Park, Suresh Mandava, Sun Young Baek, Jongkook Lee,* Collision-induced dissociation pathways of H1-antihistamines by electrospray ionization quadrupole time-of-flight mass spectrometry, Arch. Pharm. Res. 2017, 40, 736–745. (2017-06)

26.       Suresh Mandava, Bogonda Ganganna, Jungjoong Hwang, Younchang Jang, Jiho Hwang, Mallesham Samala, Ki-Bbeum Kim, Haeil Park, Ji Hyun Lee, Sun Young Baek, Jongkook Lee,* Synthesis and structure revision of dimeric tadalafil analogue adulterants in dietary supplements, Chem. Pharm. Bull. 2017, 65, 498–503. (2017-05)

27.       Han Na Park, Ji Hyun Lee, Sung-Kwan Park, Jongkook Lee,* Sun Young Baek,* Identification of a new tadalafil analogue in commercial dietary supplements: isopropylnortadalafil. Food Addit. Contam. Part A Chem. Anal. Control Expo. Risk Assess. 2017, 34, 162–169. (2017-02)

28.       Yuanying Fang, Zunhua Yang, Shankariah Gundeti, Jongkook Lee, Haeil Park,* Novel 5-nitropyrimidine derivatives bearing endo-azabicyclic alcohols/amines as potent GPR119 agonists. Bioorg. Med. Chem. 2017, 25, 254–260. (2017-01-01)

29.        Ji Hyun Lee, Han Na Park, Tan-Soon Leem, Joo-hyoung Jeon, Sooyeul Cho, Jongkook Lee,* Sun Young Baek,* Identification of new synthetic cannabinoid analogue APINAC (adamantan-1-yl 1-pentyl-1H-indazole-3-carboxylate) with other synthetic cannabinoid MDMB(N)-Bz-F in illegal products. Forensic Toxicol. 2017, 35, 45–55. (2017-01)

30.         Song Yi Lee, Jeong-Jun Lee, Ju-Hwan Park, Jae-Young Lee, Seung-Hak Ko, Jae-Seong Shim, Jongkook Lee, Moon Young Heo, Dae-Duk Kim, Hyun-Jong Cho,* Electrosprayed nanocomposites based on hyaluronic acid derivative and Soluplus for tumor-targeted drug delivery. Colloids Surf. B Biointerfaces, 2016, 145, 267–274. (2016-09-01)

31.        Ju Hee Lee, Hae Ju Ko, Eun-Rhan Woo, Sang Kook Lee, Bong Soo Moon, Chan Woo Lee, Suresh Mandava, Mallesham Samala, Jongkook Lee, Hyun Pyo Kim,*  Moracin M inhibits airway inflammation by interrupting the JNK/c-Jun and NF-κB pathways in vitro and in vivo. Eur. J. Pharmacol. 2016, 783, 64–72. (2016-07-15)

32.         Shankariah Gundeti, Jongkook Lee, Haeil Park,* Novel 1,2,3-Triazole Analogs of Sitagliptin as DPP4 Inhibitors. Bull. Korean Chem. Soc. 2016, 37, 1156–1158. (2016-07-08)

33.        Ji Hyun Lee, Han Na Park, Bogonda Ganganna, Ji Hye Jeong, Sung-Kwan Park, Jongkook Lee,* Sun Young Baek,* Isolation and structural elucidation of a new tadalafil analogue in health supplements: bisprenortadalafil. Food Addit. Contam. Part A Chem. Anal. Control Expo. Risk Assess. 2016, 33, 945–952. (2016-07)

34.     Hyeonjeong Choe, Thuy Trang Pham, Joo Yun Lee, Muhammad Latif, Haeil Park, Young Kee Kang,* and Jongkook Lee,* Remote Stereoinductive Intramolecular Nitrile Oxide Cycloaddition: Asymmetric Total Synthesis and Structure Revision of (–)-11b-Hydroxycurvularin. J. Org. Chem. 2016, 81, 2612–2617. (2016-03-18)

35.        Dong Chul Kim, Kyeong Ryang Park, Yeon Ji Jeong, Hyonok Yoon, Mi-Jeong Ahn, Gyu-Jin Rho, Jongkook Lee, Young-dae Gong, Sun-Young Han,* Resistance to the c-Met inhibitor KRC-108 induces the epithelial transition of gastric cancer cells. Oncol. Lett. 2016, 11, 991–997. (2016-02).

36.       Ji Hyun Lee, Hyung Joo Kim, Suresh Mandava, Jungjoong Hwang, Hyoung Joon Park, Sooyeul Cho, Sun Young Baek, Jongkook Lee,* Identification of a new tadalafil analogue in an adulterated dietary supplement: trans-Bisprehomotadalafil. J. Pharm. Biomed. Anal. 2015, 115, 352–358. (2015-11-08)

37.          Hye Jin Chung, Kyeong Ryang Park, Hyo Jeong Lee, Jongkook Lee, Jeong-Hyun Kim, Yong-Chul Kim, Sun-Young Han, Effects of KRC-108 on the Aurora A activity and growth of colorectal cancer cells, Biochem. Biophys. Res. Commun. 2015, 461, 605–611. (2015-07-12) 

38.     Muhammad Latif, Jeong In Yun, Kalapati Seshadri, Hyoung Rae Kim, Chi Hoon Park, Haeil Park, Hyoungsu Kim, Jongkook Lee,* Stereoselective Construction of 2,6-cis-Disubstituted Tetrahydropyrans via Intramolecular Amide Enolate Alkylation: Total Synthesis of (–)-Centrolobine. J. Org. Chem. 2015, 80, 3315–3320. (2015-03-20)

39.       Bo-Ra Lee, Sun-Young Chang, Eun-Hye Hong, Bo-Eun Kwon, Hong Min Kim, Yeon-Jeong Kim, Jongkook Lee, Hyun-Jong Cho, Jae-Hee Cheon, Hyun-Jeong Ko,* Elevated endoplasmic reticulum stress reinforced immunosuppression in the tumor microenvironment via myeloid-derived suppressor cells. Oncotarget, 2014, 5, 12331–12345. (2014-12-15)

40.         Hye Jin Chung, Majid Rasool Kamli, Hyo Jeong Lee, Jae Du Ha, Sung Yun Cho, Jongkook Lee, Jae Yang Kong, Sun-Young Han,* Discovery of quinolinone derivatives as potent FLT3 inhibitors. Biochem. Biophys. Res. Commun. 2014, 445, 561–565. (2014-03-14)

41.        Hee Sook Lee, Dae Gyu Kim, Young Sun Oh, Nam Hoon Kwon, Jin Young Lee, Doyeun Kim, Song‑Hwa Park, Jong‑Hwan Song, Sunkyung Lee, Jung Min Han, Bum‑Joon Park, Jongkook Lee, Sunghoon Kim,* Chemical suppression of an oncogenic splicing variant of AIMP2 induces tumour regression. Biochem. J. 2013, 454, 411–416. (2013-09-15)

42.         Sang-Won Hong, Kyung Hee Jung, Hee-Seung Lee, Mi Kwon Son, Hong Hua Yan, Nam Sook Kang, Jongkook Lee, Soon-Sun Hong,* SB365, Pulsatilla saponin D, targets c-Met and exerts antiangiogenic and antitumor activities. Carcinogenesis, 2013, 34, 2156–2169. (2013-09-01)

43.       Gildon Choi,¶ Jongkook Lee,¶ Jeong Yeon Ji, Jimin Woo, Nam Sook Kang, Sung Yun Cho, Hyoung Rae Kim, Jae Du Ha, Sun-Young Han,* Discovery of a potent small molecule SIRT1/2 inhibitor with anticancer effects. Int. J. Oncol. 2013, 43, 1205–1211. (2013-07-23)

44.       Sang-Won Hong, Kyung-Hee Jung, Byung Hee Park, Hong-Mei Zheng, Hee-Seung Lee, Myung-Joo Choi, Jeong In Yun, Nam Sook Kang, Jongkook Lee,* Soon-Sun Hong,* KRC-408, a novel c-Met inhibitor, suppresses cell proliferation and angiogenesis of gastric cancer. Cancer Lett. 2013, 332, 74–82.  (2013-05-10)

45.         Byung Hee Park, Kyung Hee Jung, Sun-Mi Yun, Sang-Won Hong, Jae Wook Ryu, Heejung Jung, Jae Du Ha, Jongkook Lee,* Soon-Sun Hong,* KRC-327, a selective novel inhibitor of c-Met receptor tyrosine kinase with anticancer activity. Cancer Lett. 2013, 331, 158–166. (2013-05-01)

46.      Zunhua Yang, Yuanying Fang, Tuan-Anh N. Pham, Jongkook Lee, Haeil Park, Synthesis and biological evaluation of 5-nitropyrimidine analogs with azabicyclic substituents as GPR119 agonists. Bioorg. Med. Chem. Lett. 2013, 23, 1519–1521. (2013-03-01)

47.      Tuan-Anh N. Pham, Zunhua Yang, Yuanying Fang, Jun Luo, Jongkook Lee, Haeil Park, Synthesis and biological evaluation of novel 2,4-disubstituted quinazoline analogues as GPR119 agonists. Bioorg. Med. Chem. 2013, 21, 1349–1356. (2013-03-01)

48.        Sun H. Lee, Jongkook Lee, Myung H. Jung, You M. Lee, Glyceollins, a novel class of soy phytoalexins, inhibit angiogenesis by blocking the VEGF and bFGF signaling pathways. Mol. Nutr. Food Res. 2013, 57, 225–234. (2013-02)

49.       Jeong In Yun, Hyoung Rae Kim, Haeil Park, Sang Kyum Kim, and Jongkook Lee,* Small Molecule Inhibitors of the Hedgehog Signaling Pathway for the Treatment of Cancer. Arch. Pharm. Res. 2012, 35, 1317–1333. (2012-08-31)

50.         Jongkook Lee, Sun-Young Han, Heejung Jung, Jeon Yang, Jie-Won Choi, Chong Hack Chae, Chi Hoon Park, Sang Un Choi, Kwangho Lee, Jae Du Ha, Chong Ock Lee, Jae Wook Ryu, Hyoung Rae Kim, Jong Sung Koh, Sung Yun Cho,* Synthesis and structure–activity relationship of aminopyridines with substituted benzoxazoles as c-Met kinase inhibitors. Bioorg. Med. Chem. Lett. 2012, 22, 4044–4048. (2012-06-15)

51.        Sun-Young Han, Jie Won Choi, Jeon Yang, Chong Hack Chae, Jongkook Lee, Heejung Jung, Kwangho Lee, Jae Du Ha, Hyoung Rae Kim, Sung Yun Cho,* Design and synthesis of 3-(4,5,6,7-tetrahydro-3H-imidazo[4,5-c]pyridin-2-yl)-1H-quinolin-2-ones as VEGFR-2 kinase inhibitors. Bioorg. Med. Chem. Lett. 2012, 22, 2837–2842. (2012-04-15)

52.      Sun-Young Han, Chong Ock Lee, Sung-Hoon Ahn, Mi-Ok Lee, So-Young Kang, Hyuk-Jin Cha, Sung Yun Cho, Jae Du Ha, Jae Wook Ryu, Heejung Jung, Hyoung Rae Kim, Jong Sung Koh, Jongkook Lee,* Evaluation of a Multi-kinase Inhibitor KRC-108 as an Anti-tumor Agent in Vitro and in Vivo.  Invest. New Drugs 2012, 30, 518–523. (2012-04-30)

53.       Jeong In Yun, Hyoung Rae Kim, Sang Kyum Kim, Deukjoon Kim, Jongkook Lee,* Cross-metathesis of allyl halides with olefins bearing amide and ester groups. Tetrahedron 2012, 68, 1177–1184. (2012-1-28)

54.         Jae Wook Ryu, Sun-Young Han, Jeong In Yun, Sang-Un Choi, Heejung Jung, Jae Du Ha, Sung Yun Cho, Chong Ock Lee, Nam Sook Kang, Jong Sung Koh, Hyoung Rae Kim, Jongkook Lee,* Design and synthesis of triazolopyridazines substituted with methylisoquinolinone as selective c-Met kinase inhibitors.  Bioorg. Med. Chem. Lett. 2011, 21, 7185–7188. (2011-12-1) 

55.        Tae-Gyu Nam, Jongkook Lee, John R. Walker, Achim Brinker, Charles Y. Cho, Peter G. Schultz,* Identification and Characterization of Small-Molecule Inducers of Fetal Hemoglobin. ChemMedChem  2011, 6, 777–780.  (2011-05-02)

56.         Jongkook Lee, Seung-Mann Paek, Sun-Young Han,* FMS-like tyrosine kinase 3 inhibitors: a patent review, Expert. Opin. Ther. Pat. 2011, 21, 483–503. (2011-04-30) 

57.         Jeong In Yun, Deukjoon Kim, Jongkook Lee,* Cross-metathesis of allyl halides with olefins bearing an a-alkoxy amide group. Tetrahedron Lett. 2011, 52, 1928–1930. (2011-4-20)

58.      Byungsook Kim, Te-ik Sohn, Sanghee Kim, Deukjoon Kim,* Jongkook Lee, Concise Substrate-Controlled Asymmetric Total Synthesis of (+)-3-(Z)-Dihydrorhodophytin.  Heterocycles  2011, 82, 1113–1118. (2011-2-28)

59.         Sung Yun Cho, Sun-Young Han, Chong Ock Lee, Jae Wook Ryu, Heejung Jung, Jae Du Ha, Namsook Kang, Hyoung Rae Kim, Jong Sung Koh, Jongkook Lee,* Discovery of aminopyridines substituted with benzoxazole as orally active c-Met kinase inhibitors. Bioorg. Med. Chem. Lett. 2010, 20, 4223–4227. (2010-7-15)

60.       Jongkook Lee, Jiyong Hong, Tae-Gyu Nam, Eric C. Peters, Anthony P. Orth, Bernhard H. Geierstanger, Lawrence E. Goldfinger, Mark H. Ginsberg, Charles Y. Cho, Peter G. Schultz,* A Small Molecule Inhibitor of a4 Integrin-Dependent Cell Migration.  Bioorg. Med. Chem. 2009, 17, 977–980 (Special Issue for Prof. J. A. Ellman). (2009-2-1) 

61.       Lubica Supekova, Frantisek Supek, Jongkook Lee, Shawn Chen, Nathanael Gray,  John P. Pezacki, Peter G. Schultz,* Identification of human kinases involved in hepatitis C virus replication by small interference RNA library screening.  J. Biol. Chem. 2008, 283, 29–36. (2008-1-4)

62.       Jongkook Lee, Xu Wu, Marina Pasca di Magliano, Eric C. Peters, Yan Wang, Jiyong Hong, Metthias Hebrok, Sheng Ding, Charles Y. Cho, Peter G. Schultz,* A Small-Molecule Antagonist of Sonic Hedgehog Signaling Pathway.  ChemBioChem, 2007, 8, 1916–1919. (2007-11-5)

63.       Jiyong Hong, Jongkook Lee, Kyung-Hoon Min, John R. Walker, Nathanael S. Gray, Charles Y. Cho, Peter G. Schultz,* Identification and Characterization of Small Molecule Inducers of Epidermal Keratinocyte differentiation. ACS: Chemical Biol. 2007, 2, 171-175. (2007-3-20) 

64.       Miyun Kwon, Hyun-Jin Kim, Jongkook Lee, Jaehoon Yu,* Enhanced Binding Affinity of Neomycin-Chloramphenicol (or Linezolid) Conjugates to A-Site Model of 16S Ribosomal RNA. Bull. Korean Chem. Soc. 2006, 27, 1664–1666. (2006-10-27)

65.         Jongkook Lee,* Jiyong Hong, First Synthesis and Structural Elucidation of (-)-Presphaerene. J. Org. Chem. 2004, 69, 6433–6440. (2004-9-17)

66.       Sun-Young Jang, Young Hwan Ha, Seung Whan Ko, Wonku Lee, Jongkook Lee, Sunghoon Kim, Yong Woo Kim, Won Koo Lee* and Hyun-Joon Ha,* Synthesis and antibacterial activity of arylpiperazinyl oxazolidinones with diversification of the N-substituents.  Bioorg. Med. Chem. Lett. 2004, 14, 3881–3883. (2004-8-2)

67.        Jongkook Lee, Miyun Kwon, Kyoung Hyun Lee, Sunjoo Jeong, Soon-Sil Hyun, Kye Jung Shin and  Jaehoon Yu,* An Approach to Enhance Specificity Against RNA Targets Using Hetero-Dimeric Conjugates of Aminoglycosides and Chloramphenicol (or Linezolid). J. Am. Chem. Soc. 2004, 126, 1956–1957. (2004-2-25)

68.        Hyunil Jo, Jongkook Lee, Hyoungsu Kim, Sanghee Kim and Deukjoon Kim,* Efficient construction of bicyclic system by internal SN2’ enolate alkylation/ring-closing metathesis (RCM) strategy: a concise synthesis of trans-hydrindane nucleus. Tetrahedron Lett. 2003, 44, 7043–7044. (2003-9-8)

69.      Deukjoon Kim,* Jongkook Lee, Phil Jong Shim, Joong Inn Lim, Takauki Doi and Sanghee Kim, Role of Conformational Effects on the Regioselectivity of Macrocyclic INOC Reactions: Two New Asymmetric Total Synthesis of (+)-Brefeldin A. J. Org. Chem. 2002, 67, 772–781. (2002-2-8)

70.       Deukjoon Kim,* Jongkook Lee, Phil Jong Shim, Joong Inn Lim, Hyunil Jo, and Sanghee Kim. Asymmetric Total Synthesis of (+)-Brefeldin A from (S)-Lactate by Triple Chirality Transfer Process and Nitrile Oxide Cycloaddition, J. Org. Chem. 2002, 67, 764–771. (2002-2-8)

71.    Deukjoon Kim,* Jongkook Lee, Jiyoung Chang and Sanghee Kim, Stereoselective synthesis of (±)-b-elemene by a doubly diastereodifferentiating internal alkylation: a remarkable difference in the rate of enolization between syn- and anti-esters. Tetrahedron 2001, 57, 1247–1252. (2001-2-11)

72.    Deukjoon Kim,* Phil Jong Shim, Jongkook Lee, Cheol Won Park, Sung Woo Hong, and Sanghee Kim, Construction of the Tricyclo[5.3.1.01,5]undecane System by a Novel Tandem Pinacol Rearrangement-Ene Strategy: A Formal Total Synthesis of (±)-Perhydrohistrionicotoxin. J. Org. Chem. 2000, 65, 4864–4870. (2000-7-14)

1.     “베레젠 및 플리작 허가를 바탕으로 한 2016년 미국 FDA 식물의약품 가이드라인에 대한 고찰 A Review on the 2016 US FDA Botanical Drug Development Guideline Based on Approvals of Veregen and Fulyzaq”, Insuk Song, Jungjoong Hwang, Jongkook Lee* Yakhakhoeji 2018, 62, 419–423. (2018-12-01)

2.    “세균의 Peptide Deformylase(PDF)를 억제하는 새로운 항균물질의 스크리닝 Screening of New Antibiotics Inhibiting Bacterial Peptide Deformylase (PDF)”, Jin-Hwan Kwak,* Hyunjoo Kim, Minjung Sul, Byungsun Seo, Jongkook Lee, Sooyoung Choi, Yakhakhoeji 2003, 47, 184–189. (2003-5-30)