Most Recent Publications

M. Borgini, Q. Huang, P. Chen, S. J. Geib, K. N. Houk, P. Wipf, Rhodium(I)-Catalyzed Annulation of Bicyclo[1.1.0]butyl-Substituted Dihydroquinolines and Dihydropyridines, JACS, Article ASAP, DOI: 10.1021/jacs.4c04081 Link

M. Borgini, Ł. Wieteska, C.S. Hinck, T. Krzysiak, A.P. Hinck, P. Wipf. Synthesis of 13C-methyl-labeled amino acids and their incorporation into proteins in mammalian cells. Org Biomol Chem. 2023, 21(46), 9216-9229. Link 

M. Borgini, P. Wipf. Synthesis and Rhodium(I)-Catalyzed Annulative Cleavage of Bicyclo[1.1.0]butyl Dihydroquinolines and Dihydropyridines, ChemRxiv, 2023, DOI: 10.26434/chemrxiv-2023-rnqhm. Link 

M. Borgini, P. Wipf. Synthesis of Veliparib Prodrugs and Determination of Drug-Release-Dependent PARP-1 Inhibition, ACS Medicinal Chemistry Letters, 2023, 14(5), 652-657. Link 

M. Borgini, P. Wipf. Stereoselective synthesis of δ-fluorinated isoleucines exploiting consecutive C(sp3)-H bond activations, Tetrahedron, 2022, 120, 132876. Special issue in Honor of Dr. Franziska Schoenebeck. Link 

M. Borgini, P. Mondal, R. Liu, P. Wipf. Chemical modulation of Kv7 potassium channels, RSC Medicinal Chemistry, 2021, 12, 483-537. Link 

M. Borgini, C. Zamperini, F. Poggialini, L. Ferrante, V. Summa, M. Botta, R. Di Fabio. Synthesis and Antiproliferative Activity of Nitric Oxide-Donor Largazole Prodrugs, ACS Medicinal Chemistry Letters, 2020, 11(5), 846-851. Link 

F. Orofino, G. I. Truglio, D. Fiorucci, I. D'Agostino, M. Borgini, F. Poggialini, C. Zamperini, E. Dreassi, L. Maccari, R. Torelli, C. Martini, M. Bernabei, J. F. Meis, N. K. Khandelwal, R. Prasad, M. Sanguinetti, F. Bugli, M. Botta. In vitro characterization, ADME analysis, and histological and toxicological evaluation of BM1, a macrocyclic amidinourea active against azole-resistant Candida strains, International Journal of Antimicrobial Agents, 2020, 55(3), 105865. Link 

M. Borgini, F. Orofino, G. I. Truglio, L. Balestri, M. Botta. A gram-scale synthesis of a macrocyclic amidinourea with strong antifungal activity through a Fukuyama tri-protected polyamine intermediate, Arkivoc, 2019, 4, 168- 177. Special issue in Honor of Dr. Stephen Hanessian. Link 

Brai, S. Ronzini, V. Riva, L. Botta, C. Zamperini, M. Borgini, C. I. Trivisani, A. Garbelli, C. Pennisi, A. Boccuto, F. Saladini, M. Zazzi, Maga, M. Botta. Synthesis and Antiviral Activity of Novel 1,3,4-Thiadiazole Inhibitors of DDX3X, Molecules, 2019, 24(21), 3988. Link