2021 - 2025

<2024>

54. Development of Synthetic Route for 3-Amino-5-halo-2-iodobenzoates: Versatile Starting Materials in Pharmaceutical Synthesis 

Park, Jinjae; Seo, Ju-Ahn; Cheon, Cheol-Hong

Asian Journal of Organic Chemistry, 2024, 13, e202400027. [link] 



53. Recent Progress Toward Total Syntheses of Iheyamines A and B  

Kim, Taelyn; Jeon, Jiye; Lee, Yongho; Cheon, Cheol-Hong

Asian Journal of Organic Chemistry, 2024, 13, e202300513. [link] 



52. Synthesis of a Piancol Boronate Precursor for [18F]Rucaparib Radiosynthesis 

Seo, Ju-Ahn; Park, Jinjae; Cheon, Cheol-Hong

Asian Journal of Organic Chemistry, 2024, 13, e202300501. [link] 



51. Synthesis of All Regioisomers of 2-Aryl Azaindole-3-acetic Acid Derivatives

Kim, Taewook; Park, Ju-Hyeon; Jeong, Cheol; Park, Eunjoon; Kim, Jong  Mu; Kim, You-Jin; Heo, Jung-Nyoung; Cheon, Cheol-Hong

Synthesis, 2024, 56, 860-870. [link] 



<2023>

50. Total Syntheses of 2,2’-Biindolyl Alkaloids via Cyanide-catalyzed Imino-Stetter Reaction

Park, Jinjae; Kim, Taelyn; Cheon, Cheol-Hong

Synlett, 2023, 34, 2351-2360. [link] 

(Invited Account in a Special Issue dedicated to Professor Hisashi Yamamoto on the occasion of his 80th birthday )


49. Synthesis of 2-(2-Nitrophenyl)indoline-3-acetic Acid Derivatives via Base-Catalyzed Cyclization of N-(2-Nitrobenzyl)-2-aminocinnamic Acid Derivatives

Park, Ju Hyeon; Park, Jinjae; Cheon, Cheol-Hong

Organic & Biomolecular Chemistry, 2023, 21, 1647-1652. [link] 

<2022>

48. Asymmetric Total Synthesis of Iheyamine B

Jeon, Jiye; Cheon, Cheol-Hong

Organic Letters, 2022, 24, 7128-7133.[link]

47. A Cyanide-Catalyzed Imino-Stetter Reaction Enables the Concise Total Syntheses of Rucaparib

Park, Jinjae; Cheon, Cheol-Hong

RSC Advances, 2022, 12, 21172-21180.[link]

46. Total Synthesis of Rucaparib

Park, Jinjae; Cheon, Cheol-Hong

The Journal of Organic Chemistry, 2022, 87, 4813-4817.[link]

Selected as the most-downloaded/most-read paper in April of 2022.

Highlighted in Synfacts: Synfacts 2022, 0829. https://doi.org/10.1055/s-0041-1738224 .


<2021>

45. Total Synthesis of Hinckdentine A

Jeon, Jiye; Lee, Sang Eun; Cheon, Cheol-Hong

Organic Letters, 2021, 23, 2169-2173. [link]

44. A Stereodivergent Strategy for Total Syntheses of Antirhine Alkaloids

Park, Eunjoon; Bae, Cheolwoo; Cho, Cheon-Gyu; Cheon, Cheol-Hong

The Journal of Organic Chemistry, 2021, 86, 4497-4511. [link]

43. Remarkable Differences in Reactivity between Cyanide and NHCs in Cyclization Reactions of 4-(2-Formylphenoxy)but-2-enoate Derivatives

Park, Eunjoon;  Park, Jina; Cheon, Cheol-Hong. 

( Both authors equally contributed to this work). 

Bulletin of the Korean Chemical Society, 2021, 42, 483-485. [link] 

(Invited Article for Special Issue on Chemical Synthesis & Reaction Development).