Publications
Yi-Chen Sun, Wei-Xin Shi, Wei-Chieh Kuo, Yi-Rong Hsiang, Wei-Lin Lo, Liang-Cheng Chen, Shiou-Shiow Farn, Ya-Fan Lin*, and Kuo-Ting Chen*, "Cyanopyridoimidazole/1,2-Aminothiol Click Reaction: A Novel Bioorthogonal Reaction for Synthesis of Radiotracers." Bioconjugate Chem. 2024, 35, 1, 107-114.
Shih-Chuan Tsai, Shiou-Shiow Farn, Wei-Lin Lo, Fang-Yu Ou Yang, Yong-Ching Kang, Liang-Cheng Chen, Kuo-Ting Chen, Jiunn-Wang Liao, Jui-Yin Kung, Jenn-Tzong Chen, Feng-Yun J. Huang*, "Evaluation of Chelator-to-Antibody Ratio on Development of 89Zr-iPET Tracer for Imaging of PD-L1 Expression on Tumor." Int. J. Mol. Sci. 2023, 24, 17132.
Chen KT*, "Novel Imaging Probes: From Design to Applications." Pharmaceuticals 2023, 16, 1506.
Hsu YJ, Shi WX, Tseng YC, Chiu TH, Cheng MH, Chen KT*, "Facile synthesis and anticancer activity of tetrazolyl-benzothiazole derivatives." J. Heterocycl. Chem. 2023, 60(12), 2036.
Chen KT*, Seimbille Y. "New Developments in Carbonic Anhydrase IX-Targeted Fluorescence and Nuclear Imaging Agents." Int. J. Mol. Sci. 2022, 23(11), 6125
Handula M, Verhoeven M, Chen KT, Haeck J, de Jong M, Dalm SU, Seimbille Y. “Towards Complete Tumor Resection: Novel Dual-Modality Probes for Improved Image-Guided Surgery of GRPR-Expressing Prostate Cancer.” Pharmaceutics 2022, 14, 195.
Guo CW†, Chen KT†, You TY, Lin CC, Cheng WC, “Synthesis and Evaluation of Diverse N-Substituted Disaccharide Dipeptides for Human NOD2 Stimulation Activity.” Chem. Asian J. 2022, 17, e202101169. (†Co-first authors)
Handula M, Chen KT, Seimbille Y, “IEDDA: An Attractive Bioorthogonal Reaction for Biomedical Applications Molecules”, Molecules 2021, 26(15), 4640.
Chen KT, Nieuwenhuizen J, Handula M, Seimbille Y, “A Novel Clickable MSAP Agent for Dual Fluorescence/Nuclear Labeling of Biovectors”, Org. Biomol. Chem. 2020, 18, 6134-6139
Chen KT, Nguyen K, Ieritano C, Gao F, Seimbille Y, “A Flexible Synthesis of 68Ga-Labeled Carbonic Anhydrase IX (CAIX)-Targeted Molecules via CBT/1,2-Aminothiol Click Reaction.” Molecules 2019, 24(1), 23.
Gao F, Ieritano C, Chen KT, Dias GM, Rousseau J, Bénard F, Seimbille Y, “Two bifunctional desferrioxamine chelators for bioorthogonal labeling of biovectors with zirconium-89.” Org Biomol Chem. 2018, 16, 5102-5106.
Chen KT, Ieritano C, Seimbille Y, “Early-Stage Incorporation Strategy for Regioselective Labeling of Peptides using the 2-Cyanobenzothiazole/1,2-Aminothiol Bioorthogonal Click Reaction.” ChemistryOpen, 2018, 7, 256-26.
Chen KT, Lin CK, Guo CW, Chang YF, Hu CM, Lin HH, Lai YT, Cheng TJR, Cheng WC, “Effect of the lipid II sugar moiety on bacterial transglycosylase: the 4-hydroxy epimer of lipid II is a TGase inhibitor” Chemical Communications, 2017, 53, 771-774.
Chen KT, Chen PT, Lin CK, Huang LY, Hu CM, Chang YF, Hsu HT, Cheng TJR, Wu YT and Cheng WC, “Structural Investigation of Park’s Nucleotide on Bacterial Translocase MraY: Discovery of Unexpected MraY Inhibitors” Scientific Reports, 2016, 6, 31579.
Chen KT, Huang DY, Chiu CH, Lin WW, Liang PH, Cheng WC, “Synthesis of Diverse N-Substituted Muramyl Dipeptide Derivatives and Their Use in a Study of Human NOD2 Stimulation Activity”, Chemistry-a European Journal, 2015, 21, 11984-11988.
Lin CK, Chen KT, Hu CM, Yun WY, Cheng WC, “Synthesis of 1-C-Glycoside-Linked Lipid II Analogues Toward Bacterial Transglycosylase Inhibition.”, Chemistry-a European Journal, 2015, 21, 7511-7519.
Chen KT, Kuan YC, Fu WC, Liang PH, Cheng TJ, Wong CH, Cheng WC, “Rapid preparation of mycobacterium N-glycolyl Lipid I and Lipid II derivatives: a biocatalytic approach.”, Chemistry-a European Journal, 2013, 19, 834-838.
Shih HW, Chen KT, Cheng WC, “One-pot synthesis of phosphate diesters and phosphonate monoesters via a combination of microwave-CCl3CN–pyridine coupling conditions.” Tetrahedron Letters, 2012, 53, 243-246.
Shih HW, Chen KT, Cheng TJ, Wong CH, Cheng WC, “A New Synthetic Approach toward Bacterial Transglycosylase Substrates, Lipid II and Lipid IV.”, Organic Letters, 2011, 13, 4600-4603.
Meng FC, Chen KT, Huang LY, Shih HW, Chang HH, Nien FY, Liang PH, Cheng TJ, Wong CH, Cheng WC, “Total Synthesis of Polyprenyl N-Glycolyl Lipid II as a Mycobacterial Transglycosylase Substrate.”, Organic Letters, 2011, 13, 5306-5309.
Cheng TJ, Wu YT, Yang ST, Lo KH, Chen SK, Chen YH, Huang WI, Yuan CH, Guo CW, Huang LY, Chen KT, Shih HW, Cheng YS, Cheng WC, Wong CH, “High-throughput identification of antibacterials against methicillin-resistant Staphylococcus aureus (MRSA) and the transglycosylase.”, Bioorganic & medicinal chemistry, 2010, 18, 8512-8529.
Shih HW, Chen KT, Chen SK, Huang CY, Cheng TJ, Ma C, Wong CH, Cheng WC, “Combinatorial approach toward synthesis of small molecule libraries as bacterial transglycosylase inhibitors.”, Organic & biomolecular chemistry, 2010, 8, 2586-2593.
Chen KT, Lee TW, Lo JM*, “In vivo examination of 188Re(I)-tricarbonyl-labeled trastuzumab to target HER2-overexpressing breast cancer”, Nuclear Medicine and Biology, 2009, 36, 355–361.
Chen WJ, Yen CL, Lo ST, Chen KT, Lo JM*, “Direct 99mTc labeling of Herceptin (trastuzumab) by 99mTc(I) tricarbonyl ion”, Applied Radiation and Isotopes, 2008, 66, 340-345.