Research & Professional Achievements
Research & Professional Achievements
My research focuses on the design and synthesis of targeted small molecules and bifunctional conjugates for cancer therapy, integrating synthetic chemistry with biological evaluation.
Leonidis, G.; Sigala, I.; Spathakis, M.; Kolios, G.; Giannakouros, T.; Nikolakaki, E.; Sarli, V. Synthesis of Novel SRPK1-Targeting Hybrid Compounds Incorporating Antimetabolites for Cancer Therapy. RSC. Med. Chem. 2025, 16 (12), 6285-6298.
Leonidis, G.; Koukiali, A.; Sigala, I.; Tsimaratou, K.; Beis, D.; Giannakouros, T.; Nikolakaki, E.; Sarli, V. Synthesis and Anti-Angiogenic Activity of Novel c(RGDyK) Peptide-Based JH-VII-139-1 Conjugates. Pharmaceutics 2023, 15, 381.
Chatzisideri, T.; Leonidis, G.; Karampelas, T.; Skavatsou, E.; Valentza-Almpani, A.; Bianchini, F.; Tamvakopoulos, C.; Sarli, V. Integrin-Mediated Targeted Cancer Therapy Using c(RGDyK)-Based Conjugates of Gemcitabine. J. Med. Chem 2021, 65, 271–284.